I-5900 Ingenol 3-Angelate, >99%

Synonyms : [3-Angeloyl Ingenol] [3-Angelyl Ingenol] [3-Ingenyl Angelate] [Ingenyl 3-Angelate]] [Ingenol Mebutate] [PEP005]

Related Terms : [Picato]

  • Size
  • US $
  • £
  • ¥
  • 1 mg
  • 63
  • 56
  • 43
  • 7,000
  • Add to Cart
  • Out of stock
  • 5 mg
  • 196
  • 176
  • 134
  • 21,700
  • Add to Cart
  • Out of stock
  • 10 mg
  • 332
  • 298
  • 227
  • 36,800
  • Add to Cart
  • Out of stock
  • 25 mg
  • 565
  • 507
  • 386
  • 62,700
  • Add to Cart
  • Out of stock
  • 50 mg
  • 884
  • 793
  • 604
  • 98,100
  • Add to Cart
  • Out of stock
  • 100 mg
  • 1,540
  • 1,382
  • 1,053
  • 170,800
  • Add to Cart
  • Out of stock

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  • M.W. 430.53
  • C25H34O6
  • [75567-37-2]

Special Hazard: TUMOR PROMOTER. Gloves and mask should be worn when using this compound. Care must be taken to prevent contact through all routes of exposure.

Storage: Store at or below -20 ºC. Solubility: Soluble in DMSO or ethanol. Disposal: A.

  • Protein Kinase C activator; anti-cancer drug. Hampson, P., et al. "PEP005, a selective small-molecule activator of protein kinase C, has potent antileukemic activity mediated via the delta isoform of PKC." Blood 106: 1362-1368 (2005). Kedei, N., et al. "Characterization of the interaction of ingenol 3-angelate with protein kinase C." Cancer Res. 64: 3243-3255 (2004).
  • Treatment with acids or bases or heating may cause rearrangement of the angeloyl group to the 5- or 20-positions leading to a significant decrease in potency.
  • Ingenol 3-angelate, also known as Ingenol mebutate, is the active ingredient in the drug product sold under the trade name Picato®. This drug is currently approved in at least one country for use in patients with actinic keratoses. THE INGENOL 3-ANGELATE RESEARCH COMPOUND SOLD BY LC LABORATORIES IS NOT PICATO®, AND IS NOT FOR HUMAN USE.
  • Sold for laboratory or manufacturing purposes only; not for human, medical, veterinary, food, or household use.
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